Vinca Rosea muujinta Vincriristaine
Vinga Rosea Tooska waxaa loola jeedaa Vincritine-ka dawooyinka, kaas oo laga soo qaatay Periwus-ka Periaks (Vingascar Periwinks, oo loo yaqaan 'periwinklor', oo ah periwink-ka, waa noocyada perifle, waa noocyo unugyo ah oo dhirta ubax ah Qoyska Apococynaceeae.
Vincritine waa alkaloid dabiici ah oo loo istcimaalo daaweynta kemotherabi ee lagu daaweeyo noocyo kala duwan oo kansarka, oo ay ku jiraan Thuukemia, limboon, iyo burooyinka adag. Waxay ka shaqaysaa iyada oo carqaladeynaysa koritaanka unugyada kansarka.
Waxyaabaha ugu muhiimsan ee firfircoon ee Shiinaha | Magaca Ingiriisiga | CAS MAYA. | Miisaanka Moleculal | Qaaciddada molika |
长春胺 | Vamine | 1617-90-9 | 354.44 | C21h26n2O3 |
脱水长春碱 | Anhydrovinblateine | 38390-45-3 | 792.96 | C46h56n4o8 |
異長春花苷內酰胺 | Stricosamide | 23141-25-5 | 498.53 | C26H30N2O8 |
四氢鸭脚木碱 | Tetrahdrodronalstone | 6474-90-4 | 352.43 | C21H24N2O3 |
酒石酸长春瑞滨 | VINORELLBE TARCRATER | 125317-39-7 | 1079.12 | C45h54n4o8.2 (c4h6o6); c |
长春瑞滨 | VINORELLINE | 71486-2-1 | 778.93 | C45h54n4o8 |
长春新碱 | Micninbine | 57-22-7 | 824.96 | C46h56n4o10 |
硫酸长春新碱 | Vincritine sulfate | 2068-78-2 | 923.04 | C46h58n4o14s |
硫酸长春质碱 | Catharanthine sulfate | 70674-90-7 | 434.51 | C21h26n2O6s |
酒石酸长春质碱 | Haydhantrate | 4168-17-6 | 486.51 | C21h24n2o2.c4h6O6 |
长春花碱 | Vinblaaste | 865-21-4 | 810.99 | C46h58n4o9 |
长春质碱 | Eegarandine | 2468-21-5 | 336.43 | C21H24N2O2 |
文朵灵 | Falwadshor | 2182-14-1 | 456.53 | C25h32n2o6 |
硫酸长春碱 | Vinblastine sulfate | 143-67-9 | 909.05 | C46h60n4o13s |
谷甾醇 谷甾醇 谷甾醇 | β-fastosterol | 83-46-5 | 414.71 | C29h50o |
菜油甾醇 | Bixidmonsto | 474-62-4 | 400.68 | C28H48O |
齐墩果酸 | Olecolom acid | 508-02-1 | 456.7 | C3h48o3 |
Faahfaahinta alaabada | ||
Magaca wax soo saarka: | Vinca Rosesea Bad | |
Magaca Botanic: | Catharanthus Roseus (L.) | |
Qayb dhirta | Ubax | |
Wadanka uu ka yimid: | Maacuun | |
Alaabada falanqaynta | Cayimid | Habka Tijaabada |
Muuqashada | Budo fiican | Digtooniya |
Midab | Budada gaagaaban | Ee aragtiyeed |
Ur & dhadhanka | Sifo | Digtooniya |
Aqoonsi | Isku mid ah muunad | Hptlc |
Saamiga soosaarka | 4: 1 ~ 20: 1; Vincritine 98% min | |
Falanqaynta talaabooyinka | 100% illaa 80 mesh | USP39 <786> |
Luminta qalajinta | ≤ 5.0% | EUR.PH.9.0 [2.5.12] |
Isugeynta ash | ≤ 5.0% | EUR.PH.9.0 [2.4.16] |
Hogaanka (PB) | ≤ 3.0 mg / kg | EUR.PH.9.0 <2.58> ICP-Ms |
Arsenic (sida) | ≤ 1.0 mg / kg | EUR.PH.9.0 <2.58> ICP-Ms |
Cadmium (CD) | ≤ 1.0 mg / kg | EUR.PH.9.0 <2.58> ICP-Ms |
Meerkuriga (hg) | ≤ 0.1 mg / kg -reg.ec629 / 2008 | EUR.PH.9.0 <2.58> ICP-Ms |
Bir culus | ≤ 10.0 mg / kg | EUR.PH.9.0 <2.4.8> |
KHATARTA KHATARTA | Waa u qalmaa euro.ph. 9.0 <5,4> iyo EC Yurub Tilmaanta Yurub 2009/32 | EUR.PH.9.0 <2.4.24> |
Hadhaagii sunta cayayaanka | Xeerar isku-dhafan (EC) No.396 / 20055/20050 Reg.2008 / 839 / CE | Korofiska gaaska |
Bakteeriyada aerobic (TAMC) | ≤10000 cfu / g | USP39 <61> |
Khamiir / caaryada (TAMC) | ≤1000 cfu / g | USP39 <61> |
Escherichia Coli: | Ka maqnaa 1g | USP39 <62> |
Salmonella SP: | Ka maqnaa 25g | USP39 <62> |
Staphylococcus aureus: | Ka maqnaa 1g | |
Listeria MonocyTogenens | Ka maqnaa 25g | |
Aflatoxins b1 | ≤ 5 ppb -reg.ec 1881/2006 | USP39 <62> |
Aflatoxs σ b1, b2, g1, g2 | ≤ 10 ppb -reg.ec 1881/2006 | USP39 <62> |
Tilmaamaha sheyga ee Vinga Rosea Vincrirista Vinchas-ka ayaa waxaa ka mid noqon kara:
Daahirsanaanta sare:Alaabada Vincritinine waxay badanaa leeyihiin daahir sare oo u hoggaansanaanta heerar adag oo wax soo saarka daroogada si loo hubiyo daahirka iyo xasilloonida daroogada.
Isha laga helo raadinta:Vincritine-ka waxaa badanaa laga soo saaraa dhirta 'Catharanthus Roseus'. Geedihiisa wax soo saarka ayaa la raadraacayaa oo waafaqsanaada iyo tilmaamaha wax soo saarka ee aruurinta iyo wax soo saarka ee qalabka dawooyinka botanical.
Deganaanshaha kiimikada:Sida xarunta alkaloid, Vincritine waxay leedahay xasillooni kiimiko ah oo wanaagsan waxayna ku habboon tahay wax soo saarka dawooyinka iyo kaydinta muddada-dheer.
Falalka ka hortaga burada:Sida daroogada ka hortaga burada, Vincritine waxay leedahay nashaadyada xakameynta koritaanka iyo fiditaanka unugyada burooyinka waxayna ku habboon yihiin daaweynta kansarka kaladuwan.
Xaqiijinta caafimaad:Vincritine-ka si dhakhso ah ayaa loo xaqiijiyey waxaana si ballaaran loogu isticmaalaa waxqabadka caafimaadka, iyadoo la adeegsanayo takoorida xogta la isku halleyn karo iyo takhaatiirta caafimaad.
Astaamahaas badeecadan ayaa iftiiminaya tayada, nashaadaadka, iyo qiimaha caafimaad ee Vincritine-ka miccritine inay tahay daroogada ka hortagga kansarka.
Vinga Rosea oo laga soo saaro Vincrirista-ga waxaa ugu horreyn lagu yaqaanaa codsiyada dawooyinka ee daaweynta kansarka mana ahan caadi ahaan la xidhiidha dheefaha caafimaadka tooska ah ee isticmaalka macaamilka guud. Vincritine, oo ka soo baxay warshaddii Vinga Rosea, waa daawada kiimikaad ee loo yaqaan 'themotherapy chotheraprapy', uu yahay daawada kemotherapy chotheraprapy kor ku qaad ee loo isticmaalo noocyada kansarka kala duwan, oo ay ku jiraan qanjirada, qanjirada, iyo burooyinka adag. Waxay ku shaqeysaa iyada oo faragelin ku sameeya koritaanka unugyada kansarka.
Waxaa muhiim ah in la ogaado in vincritine-ka uu yahay dawooyinka dhakhtarku qoro ee lagu maareeyo kormeerka xirfad-yaqaannada daryeelka caafimaadka, oo ay la xiriiraan dhibaatooyinka soo raaca iyo halista. Sidaa darteed, caadi ahaan looma suuq geysto ama loo cuno faa'iidooyinkeeda caafimaad ee ka baxsan meelaynta caafimaad.
Codsiyada faahfaahsan ee Vinga Rosea Tooska Vincrirista Vincritine waxaa ka mid ah:
Daaweynta Kansarka:Vincritine-ka waxaa ugu horreyn lagu isticmaalaa daaweynta noocyada kala duwan ee kansarka, oo ay ku jiraan Thuukemia, Lympoma, iyo Burooyinka adag. Waxaa la qaataa iyada oo qayb ka ah daaweynta kemotherabi lagu hayo in la xakameeyo koritaanka unugyada kansarka.
Daraasad dawladeed:Soosaarka ayaa loo adeegsadaa cilmi-baarista dawooyinka ee ku saabsan horumarinta daaweynta cusub ee dawooyinka cusub iyo daraasadda habaynta ficil.
Chemistry daawo:Vincritine waxay u adeegtaa sidii xarun qiimo leh oo ku taal miyiga ee cilmiga dawooyinka, kuna biirinta horumarinta dawooyinka cusub iyo wakiillada daweynta.
Bayoolaji:Soosaarka waxaa laga yaabaa in laga shaqeeyo codsiyada bayoolajiga, sida soo saarista foomka dawooyinka lidka ku ah iyo nidaamyada gaarsiinta daroogada.
Tijaabooyinka caafimaad:Vincritine waxay ku lug leedahay tijaabooyinka caafimaad si loo sahamiyo wax ku oolnimadiisa ee lagu daweeyo noocyo kala duwan oo kansarka ah iyo in la baaro codsiyada suurtagalka ah ee xaaladaha kale ee caafimaad.
Qaadashada daroogada:Soosaarka waxaa loo isticmaalaa sameynta dawooyinka wax soo saarka dawooyinka, oo ay ku jiraan xalka lagu durey iyo foomamka kale ee daweynta kansarka.
Codsiyadan ayaa muujinaya adeegsiga kaladuwan ee Vinga Rosea ee Vingacea ee ku jira daaweynta kansarka, cilmi baarista dawooyinka, iyo horumarka daroogada.
Vincritine-ka waa daawada kemotherapy kor u qaadida kiimiko ah, oo isticmaalkiisa waxaa lala xiriiri karaa dhowr waxyeel oo suurtagal ah. Qaar ka mid ah waxyeelooyinka suurtagalka ah ee budada Vincritine waxaa ku jiri kara:
Neurotoxicity:Vincritine waxay u geysan kartaa waxyeelo nidaamka neerfaha ee go'doomin, taasoo keenta astaamaha sida kabuubyada, xirashada, iyo daciifnimada xididdada.
Saamaynta caloosha ee caloosha:Waxyeelooyinka caloosha ee caadiga ah waxaa ka mid noqon kara lallabbo, matag, calool fadhi, iyo calool xanuun.
Xadgudubka Marroo ee lafta:Vincritine waxay xakamayn kartaa dhuuxa lafta, taasoo horseedaysa wax soo saarka unugyada dhiigga, kaas oo sababi kara dhiig-yaraan, oo kor u qaadaya u nugul caabuqa, iyo hanuuninta dhiigbaxa.
Timo lumis:Shakhsiyaadka qaar waxay la kulmi karaan timo lumis ama timaha oo timaha ka dhalata daaweyn vincritine.
Jaw xanuun:Vincritine-ka waxay sababi kartaa nooc cayiman oo xanuun ah oo loo yaqaan "vincritine-ka-daadashada neuropathy-oduther-ba'an, oo lagu garto xanuunka daanka iyo liqidda oo dhib badan.
Saameynta kale ee jirta:Waxyeello kale oo soo gaaraya waxaa ka mid noqon kara daciifnimo muruqyada, isbeddelada dhiig karka, iyo xasaasiyadda xasaasiyadda.
Waxaa muhiim ah in la ogaado in liistada kor ku xusan aysan ahayn mid dhammaystiran, iyo xirfadlayaal daryeel caafimaadku waa inay si dhaw ula socdaan shakhsiyaadka ka hela Vincritine-ka wixii waxyeelo ah ee suurtagalka ah. Dhibaatooyinka gaarka ah ee dawooyinka iyo darnaantooda way ku kala duwanaan karaan qof ilaa qof. Bukaannadu waa inay ka wada hadlaan waxyeelooyinka suurtagalka ah iyo walaacyada daryeel-caafimaadeedka daryeel caafimaadkooda kahor bilaabida daaweynta vincritisteritine.
Baakadaha iyo Adeegga
Ka iibsi
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Maraakiibta
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Bixinta iyo hababka gudbinta
Muujin
100kg, 3-5 maalmood
Albaabka adeegga albaabka ayaa si fudud u soo qaadaya alaabada
By badda
In ka badan300kg, ku dhawaad 30 maalmood
Dekadda loogu talagalay Diyaaradda Xirfadlaha Adeegga Dekadda ee loo baahan yahay
Hawada
100kg-1000kg, 5-7 maalmood
Gegada Diyaaradaha ee Diyaaradda Aqalka Diyaaradaha ee Diyaaradda ayaa loo baahan yahay
Faahfaahinta Soo-Saarka (Qiyaasta qulqulka)
1. Fadhig iyo goosashada
2. Soo saarista
3. U fiirsashada iyo nadiifinta
4. Qalajinta
5. Heerka
6. Xakamaynta Tayada
7. Baakadaha 8. Qaybinta
Shahaado
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