Stephania waxay soo saartaa budada Cepharanthine

Magaca Alaabta: Stephania Japonica Extract
Asal Laatiinka: Stephania cephalantha Hayata(Stephania japonica (Thunb.)Miers
Muuqashada: Caddaan, Budada Cad Cawlan
Walaxda firfircoon: Cepharanthine 80% -99% HPLC
Qaybta la isticmaalo: Tuber/Root
Codsiga: Alaabooyinka daryeelka caafimaadka
Barta dhalaalka: 145-155°
Wareeg gaar ah: D20+277°(c=2inchloroform)
Barta karkarinta: 654.03°C (qiyaasta qallafsan)
Cufnaanta: 1.1761 (qiyaas adag)
Tusmada dib-u-celinta: 1.5300 (qiyaas)
Xaaladaha kaydinta: underinertgas (nitrogen ama argon) at2-8°C
Solubility: Ku milma SO (35mg/ml) ama ethanol (20mg/ml)
Isku-dhafka aysiidhka (pKa): 7.61 ± 0.20 (La saadaaliyay)


Faahfaahinta Alaabta

Warar Kale

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Hordhac Product

Stephania Extract Cepharanthine Powder waa walax ka soo jeeda digriiga geedka Stephania cephalantha Hayata (Stephania japonica (Thunb.) Miers) ama Stephania epigaea Lo/Stephania yunnanensis HSLo.Cepharanthine waa badeeco dabiici ah oo ka go'doonsan geedkan waxaana lagu sameeyay daraasado kala duwan sababo la xiriira sifooyinka dawooyinka ee suurtagalka ah.Waxaa la ogaaday inay muujiso waxqabadyada ka-hortagga SARS-CoV-2, taasoo muujinaysa waxtarka xakamaynta faafitaanka fayraska.Intaa waxaa dheer, Cepharanthine waxay muujisay awoodda ay u leedahay inay dib u celiso P-glycoprotein (P-gp) - dhexdhexaadinta caabbinta daawooyinka badan ee unugyada qaarkood waxayna kor u qaadaysaa dareenka wakiilada kansarka ee moodooyinka tijaabada ah.Waxaa intaa dheer, waxaa la muujiyay in ay saameyn ku leedahay beerka bini'aadamka cytochrome P450 enzymes CYP3A4, CYP2E1, iyo CYP2C9, waxayna la xiriirtaa antitumor, anti-bararka, iyo saameynta antinociceptive.
Marka la soo koobo, Stephania Extract Cepharanthine Powder waa nooc budo ah oo ka mid ah alaabta dabiiciga ah ee Cepharanthine oo ka soo jeeda dhirta Stephania cephalantha, taas oo muujisay suurtagalnimada codsiyada dawooyinka kala duwan.

Faahfaahin (COA)

Alaabta Cepharanthine
CAS 481-49-2
Qiimayn 80% ~ 99%
Muuqashada budo cad
Baakad 1KG/Bac
Shayga Tilmaamid
Muuqashada budo cad cawl, ur dhexdhexaad ah, heer sare ah hygroscopic
Aqoonsiga TLC: Xalka caadiga ah iyo tijaabada xal isku mid ah, RF
Qiimaynta (Asal qalalan) 98.0% --102.0%
Muuqaal gaar ah -2.4°~ -2.8°
PH 4.5 ~ 7.0
Biraha culus (Sida Pb) ≤10pm
As ≤1ppm
Pb ≤0.5pm
Cd ≤1ppm
Hg ≤0.1pm
Walaxda la xidhiidha Bar aan ka weynayn meesha xalinta caadiga ah
Walxaha haraaga ah <0.5%
Waxyaabaha Biyaha <2%

Tilmaamaha Alaabta

Stephania Extract Cepharanthine Powder waa badeeco dabiici ah oo laga helay geedka Stephania cephalantha Hayata.Waxaa la ogaaday in ay leedahay dhowr guri oo dawooyin ah, oo ay ku jiraan:
1. Hawlaha ka hortagga SARS-CoV-2
2. Saamaynta xannibaadda ee faafinta fayraska
3. Dib-u-noqoshada iska caabbinta dawooyinka badan ee P-glycoprotein-dhexdhexaadin
4. Kobcinta dareenka wakiilada ka hortagga kansarka
5. Saamaynta xannibaadda ee beerka cytochrome P450 enzymes CYP3A4, CYP2E1, iyo CYP2C9
6. Antitumor, anti-bararka, iyo saamaynta antinociceptive

Waa maxay biosynthesis ee Cepharanthine?

Biosynthesis of cepharanthine ee Stephania waxay ku bilaabataa uumi dopamine iyo 4-hydroxyphenylacetaldehyde (4-HPAA, 5) iyada oo loo marayo norcoclaurine synthase (NCS), taasoo keenta norcoclaurine.

Waa maxay milanka Cepharanthine?

Cepharanthine waxay ku milmi kartaa dareerayaasha organic sida ethanol, DMSO, iyo dimethyl formamide (DMF).Solubility of cepharanthine ee dareerayaashan waa qiyaastii 2, 5, iyo 10 mg/ml, siday u kala horreeyaan.Cepharanthine si yar bay ugu milmi kartaa kaydadka aqueous.

Codsiyada

Warshadaha arji ee Stephania Extract Cepharanthine Powder waxaa ka mid ah Pharmaceutical, Nutraceutical, Biotechnology, and Herbal Medicine, codsiyada ugu muhiimsan waa sida soo socota:
Isticmaalka suurtagalka ah ee daaweynta fayraska
Suuragal ahaan kaaliye ahaan daaweynta kansarka
Suurtagalnimada in loo isticmaalo daawaynta ka hortagga bararka
Macquul ah sida wakiilka xanuunka
Codsiyadani waxay muujinayaan isticmaalka kala duwan ee suurtogalka ah ee Stephania Extract Cepharanthine Powder ee noocyada kala duwan ee daaweynta.


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    * Miisaanka saafiga ah: 25kgs/ durbaan, Miisaanka Guud: 28kgs/Drum
    * Cabbirka durbaanka & mugga: ID42cm × H52cm, 0.08 m³/ durbaan
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